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Bibliografia APIS  

C. Annoni, E. Nakata, T. Tamura, F. F. Liew, S. Nakano, M. L. Gelmi, T. Morii “Construction of Ratiometric Fluorescent Sensors by Ribonucleopeptides” Org. Biomol. Chem., 2012, 10, 8767-8769.


A. Contini, G. Cappelletti, D. Cartelli, G. Fontana, M.L. Gelmi “Molecular Dynamics and Tubulin Polymerization Kinetics Study on 1,14-Heterofused Taxanes: Evidences of Stabilization of the Tubulin Head-to-Tail Dimer-Dimer Interaction” Molecular BioSystems, 2012, 8, 3254-3261


A. Ruffoni, A. Casoni, M. L. Gelmi, S. Pellegrino, F. Clerici “Hydroarylation of Substituted Norbornene Amino Acids: Studies on Long-Range Stereo-Electronic Effects on the Regioselectivity of the Addition” Current Organic Chemistry, 2012, 16, 2724-2738.


A. Contini, E. Erba, S. Pellegrino, “Multicomponent Synthesis of Pentyl-Sulfonyl Amidines via Diazoalkane” Synlett, 2012, 23, 1523-1525.


C. M. Greco, M. Camera, L. Facchinetti, M. Brambilla, S. Pellegrino, M. L. Gelmi, E. Tremoli, A. Corsini, N. Ferri, “Chemotactic effect of prorenin on human aortic smooth muscle cells: a novel function of the (pro)renin receptor” Cardiovascular research, 2012, 95, 366-374



S. Pellegrino, A. Contini, F. Clerici, A. Gori, D. Nava, M. L.  Gelmi, “1H-Azepine-4-amino-4-carboxylic acid: a new α, α disubstituted ornithine analogue capable of inducing helix conformations in short Ala-Aib pentapeptides” Chemistry- a European Journal, 2012, 1, 8705-8715


S. Pellegrino, C. Annoni, A. Contini, F. Clerici, M. L. Gelmi, “Expedient chemical synthesis of 75mer DNA binding domain of MafA: an insight on its binding to insulin enhancer” Amino Acids, 2012, 43, 1995-2003.


M. Penso, F. Foschi, S. Pellegrino, A. Testa, M. L. Gelmi, “Diastereoselective protocols for the synthesis of 2,3 trans- and 2,3 cis-methoxy-morpholine-2-carboxylic acid derivatives” J. Org. Chem. 2012, 77, 3454-3461.


A. Ruffoni, A. Casoni, S. Pellegrino, M.L. Gelmi, R. Soave, F. Clerici, “Sulfanyl-methylene-5(4H)-oxazolones and β-sulfanyl-α-nitroacrylates as appealing dienophiles for the synthesis of conformationally constrained cysteine analogues” Tetrahedron, 2012, 68, 1951-1962.


N. Ferri, T. Radice, M. Antonino, E. M. Beccalli, S. Tinelli, F. Zunino, A. Corsini, G. Pratesi, E. M. Ragg, M. L. Gelmi, A. Contini  “Synthesis, structural, and biological evaluation of bis-heteroarylmaleimides and bis-heterofused imides” Bioorg. & Med. Chem. 2011, 19, 5291-5299.


G. Lanza, U. Chiacchio, S. Motta, S. Pellegrino, G. Broggini “On the Stability of Polyalanines  Secondary Structures: the Role of Polyproline II Helix” Chem. Phys. Chem. 2011, 12, 2724-2727


F. Gassa, A. Contini, G. Fontana, S. Pellegrino, M.L. Gelmi, “A Highly Diastereoselective “Synthesis of a -Hydroxy-β -amino Acid Derivatives via a Lewis Acid Catalyzed Three-Component Condensation Reaction.”    J. Org. Chem.  2010, 75, 7099-7106.


D. Rigamonti, C. Mutti, C. Zuccato, E. Cattaneo, A. Contini “Turning REST/NRSF Dysfunction in Huntington's Disease into a Pharmaceutical Target.” Curr. Pharm. Des.2009, 15, 3958-3967


S. Pellegrino, N. Ferri, N. Colombo, E. Cremona, A. Corsini, R. Fanelli, M. L. Gelmi, C. Cabrele “Synthetic peptides containing a conserved sequence motif of the Id protein family modulate vascular smooth muscle cell phenotype” Bioorg. Med. Chem. Lett., 2009, 19, 6298–6302.


N. Ferri, A. Corsini, P. Bottino, F. Clerici, A. Contini “Virtual screening approach for the identification of new Rac1 inhibitors” J. Med. Chem. 2009, 52, 4087-4090.


S. Pellegrino, F. Clerici, M. L. Gelmi “b-Hydroxynorbornane amino acid derivatives: valuable synthons for the diastereoselective synthesis preparation of substituted cyclopentylglycines derivatives” Tetrahedron 2008, 64, 5657-566


M. L. Gelmi, F. Clerici, R. Gandolfi, S. Pellegrino “A new efficient synthesis of enantiopure diasteromeric 3’-aminocyclopentylglycines” Tetrahedron-Asymmetry 2008, 19, 584-592


S. Leone, C. Mutti, A. Katzantsev, E. Cattaneo, M. Sturlese, S. Moro, D. Rigamonti, A. Contini “SAR and QSAR Study on 2-Aminothiazole Derivatives, Modulators of Transcriptional Repression in Huntington's Disease” Bioorg. & Med. Chem. 2008, 16, 5695-5703.


N. Ferri, E. M. Beccalli, A. Contini, A. Corsini, M. Antonino, T. Radice, G. Pratesi, S. Tinelli, F. Zunino, M. L. Gelmi “Antiproliferative effects on human tumor cells and rat aortic smooth muscular cells of 2,3-heteroarylmaleimides and heterofused imides” Bioorg. & Med. Chem. 2008, 16, 1691-1701.


M. L. Gelmi, C. Cattaneo, S. Pellegrino, F. Clerici, M. Montali, C. Martini “An efficient route to all stereoisomeric enantiopure 6-amino-3-alkyl-3-azabicyclo[3.2.1]octane-6-carboxylic acids”  J. Org. Chem. 2007, 72, 9811-9814.


M. L. Gelmi, F. Caputo, F. Clerici, S. Pellegrino, G. Giannaccini, L. Betti, L. Fabbrini, L. Schmid, L. Palego, A. Lucacchini “1-Aminocyclopentane-1,2,4-tricarboxylic acids screening on glutamatergic and serotonergic systems”  Bioorg. Med. Chem., 2007, 15, 7581–7589


F.Caputo, C. Cattaneo, F. Clerici, M.L. Gelmi, S. Pellegrino “α,γ-Diamino Acids: Asymmetric Synthesis of New Constrained 6-Amino-3 azabicyclo[3.2.1] octane-6-carboxylic Acids” J. Org. Chem. 2006, 71, 8467-8472.


 F. Caputo, F. Clerici, M.L Gelmi, S. Pellegrino, D. Pocar “An efficient synthesis of new diastereomeric enantiopure 1-aminocyclopentane-1,2,4-tricarboxylic acids” Tetrahedron:Asymmetry, 2006, 17, 1430-1436.


 C. Cabrele, F. Clerici, M.L. Gelmi, R. Gandolfi, F. Molinari, S. Pellegrino “Chemoenzymatic resolution of epimeric cis 3-carboxycylopentylglycine derivatives” Tetrahedron, 2006, 62, 3502-3508


 F. Caputo, F. Clerici, M.L Gelmi, S. Pellegrino, T. Pilati  “Enantioselective Synthesis of Epimeric cis  3-Carboxycylopentylglycines” Tetrahedron:Asymmetry, 2006, 17, 61-67.


F. Caputo, F. Clerici, M. L. Gelmi, D. Nava, S. Pellegrino “Uncatalyzed Solventless Diels-Alder Reaction of 2-Amino-3-nitroacrylate: Synthesis of New Epimeric 2-Amino-3-nitro-norbornene- and norbornane-2-carboxylic Acids” Tetrahedron, 2006, 62, 1288-1294


F. Clerici, M. L. Gelmi, S. Pellegrino, T. Pilati “3-Formylcyclopent-3-enyl- and 3-carboxycyclopentylglycine Derivatives: a New Stereocontrolled Approach via Retro-aldol or Retro-Claisen Reactions” J. Org. Chem. 2003, 68, 5286.


M. L. Gelmi, D. Pocar     "Heterosubstituted carbocyclic a-amino acids. A review" Org. Prep. Proc. Int. 2003, 35, 141.


F. Clerici, M. L. Gelmi, D. Pocar, T. Pilati “Masked constrained cysteines: diastereoselective and enantioselective synthesis of 1-amino-2-mercaptocyclopropanecarboxylic acid derivatives" Tetrahedron: Asymmetry 2001, 12, 2663.


F. Clerici, A. Gambini, M. L. Gelmi, D. Nava "Carbocyclic Serine Analogues: Regio- and Diastereoselective Syntheses of New 1-Amino-2,5-Dihydroxycyclohexanecarboxylic Acids " Tetrahedron 2001, 57, 6429.


F. Clerici, A. Gambini, M. L. Gelmi "A Highly Diastereoselective Synthesis of New Polyhydroxylated 2-Aminonorbornanecarboxylic Acids" J. Org. Chem. 2001, 66, 4941.


G. Abbiati, F. Clerici, M. L. Gelmi, A. Gambini, T. Pilati    "Asymmetric Synthesis of 2-Amino-3-hydroxynorbornene-2-carboxylic Acid Derivatives" J. Org. Chem. 2001, 66, 6299.


F. Clerici, M. L. Gelmi, A. Gambini "Conformationally constrained serine analogues: synthesis of new 2-amino-3-hydroxynorbornanecarboxylic acid derivatives"

J. Org. Chem. 2000, 65, 6138.


F. Clerici, M. L. Gelmi, D. Pocar "A novel class of conformationally constrained masked cysteines: synthesis of 2-alkyl and 2-arylsulfanyl-1-aminocyclopropanecarboxylic acids"  J. Org. Chem.1999, 64, 726.


F. Clerici, M. L. Gelmi, A. Gambini "A highly diastereoselective approach to conformationally constrained serine analogues: synthesis of a a-amino-b-hydroxycyclohexenecarboxylic acid and derivatives" J. Org. Chem. 1999, 64, 5764.



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